Selective HDAC1 and HDAC2 Inhibitor
Home > PRODUCTS > Biochemicals > Selective HDAC1 and HDAC2 Inhibitor

Diversity screening library discount

Newsletter Subscription

Stay updated with our new products and services. You can unsubscribe at any time.

Selective HDAC1 and HDAC2 Inhibitor

methyl N-[[4-[[2-amino-5-(2-thienyl)phenyl]carbamoyl]phenyl]methyl]carbamate

Histone deacetylase HDAC1 inhibitor IC50 = 6 nM, HCT-116 mouse xenograft model GI50 = 100 nM


OTAVAchemicals Catalogue Number: 7070707089
CAS Registry Number: 1013330-84-1

Purity: 98%


Ref.: Witter et al. Optimization of biaryl Selective HDAC1&2 Inhibitors (SHI-1:2). Bioorganic & Medicinal Chemistry Letters (2008), 18, 726-731

Abstract: Selective HDAC1/2 inhibitor, exhibiting selectivity over class II HDACs 3–8. Histone deacetylases are considered promising targets for cancer epigenetic therapy

DOI: 10.1016/j.bmcl.2007.11.047

Price info:
1 MG 20 EUR
5 MG 70 EUR
10 MG 100 EUR
300uL of 10mM solution

35 EUR