4-oxo-1H-benzo[h]quinoline-3-carboxylic acid

 protein kinase CK2 inhibitor, IC50 = 1 µM

OTAVAchemicals Catalogue Number: 0107830116

CAS Registry Number: 35957-14-3

(CAS Registry Number: 51726-83-1)

Purity: 95% (HPLC)

Ref.: J. Med. Chem. 2006, 49, 22, 6443–6450

Abstract: It was revealed that the most active compound 4-oxo-1,4-dihydrobenzo[h]quinoline-3-carboxylic acid (IC50 = 1 µM) is ATP competitive (Ki value is 0.28 µM)

DOI: 10.1021/jm050048t