N-(6-Benzyl-2-phenethylamino-5,6,7,8-tetrahydro-pyrido[4,3-d]pyrimidin-4-yl)-3-chloro-2-methyl-benzenesulfonamide

CaMKII inhibitor

Chemical Formula: C29H30ClN5O2S

Molecular Weight: 548.1

OTAVAchemicals Catalogue Number:  7139318

CAS Registry Number:  1208123-85-6

Purity: >95%

Ref.: Bioorg Med Chem Lett. 2010 Nov 15;20(22):6696-8.

Abstract: CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM; significantly high selectivity against CaMKIV, MLCK, p38a, Akt1, and PKC. 

DOI: 10.1016/j.bmcl.2010.09.005